Umlobi: Marcus Baldwin
Usuku Lokudalwa: 17 Ujuni 2021
Ukuvuselela Usuku: 23 Ujuni 2024
Anonim
Treatment of Alzheimer’s Disease - Galantamine, Rivastigmine, and Donepezil
Ividiyo: Treatment of Alzheimer’s Disease - Galantamine, Rivastigmine, and Donepezil

-Delile

IGalantamine isetshenziselwa ukwelapha izimpawu zesifo i-Alzheimer's (AD; isifo sobuchopho esonakalisa kancane inkumbulo kanye nekhono lokucabanga, ukufunda, ukuxhumana nokuphatha imisebenzi yansuku zonke). IGalantamine isekilasini lemithi ebizwa nge-acetylcholinesterase inhibitors. Isebenza ngokwandisa inani lento ethile yemvelo ebuchosheni edingeka kwimemori nasekucabangeni. IGalantamine ingathuthukisa ikhono lokucabanga nokukhumbula noma yehlise ukulahleka kwalawa makhono kubantu abane-AD. Kodwa-ke, i-galantamine ngeke yelaphe i-AD noma ivimbele ukulahleka kwamakhono engqondo ngesikhathi esizayo.

IGalantamine iza njengethebhulethi, i-capsule ekhishwe isikhathi eside (esebenza isikhathi eside), nesisombululo (uketshezi) okufanele sithathwe ngomlomo. Amaphilisi noketshezi kuvame ukuphuzwa kabili ngosuku, okungcono ngokudla kwasekuseni nakusihlwa. Ama-capsule akhululwa enwetshiwe ngokuvamile athathwa kanye ngosuku ekuseni. Thatha i-galantamine cishe ngesikhathi esifanayo (ama) nsuku zonke. Landela izinkomba ezikulebuli kadokotela wakho ngokucophelela, bese ubuza udokotela noma usokhemisi wakho ukuthi akuchaze nganoma iyiphi ingxenye ongayiqondi. Thatha i-galantamine njengoba nje kuqondisiwe. Ungayithathi kancane noma uyithathe kaningi kunokuyalelwa ngudokotela wakho. Mancane amathuba okuthi ube nemiphumela engemihle ye-galantamine uma ulandela isheduli yokulinganisa ngqo enqunywe udokotela wakho.


Gwinya wonke amaphilisi akhishwe isikhathi eside; ungazichobozi noma uzihlafune.

IGalantamine ingacasula isisu sakho, ikakhulukazi ekuqaleni kokwelashwa kwakho. Thatha i-galantamine ngokudla uphuze izingilazi zamanzi ezi-6 kuya kwezi-8 nsuku zonke. Lokhu kunganciphisa ithuba lokuthi uzoba nesisu esibuhlungu ngesikhathi sokwelashwa kwakho.

Udokotela wakho kungenzeka akuqale ngomthamo ophansi we-galantamine futhi akhuphule kancane umthamo wakho, hhayi kaningi ngaphezu kwesisodwa njalo emavikini amane.

Qhubeka uthathe i-galantamine noma ngabe uzizwa uphilile. Ungayeki ukuthatha i-galantamine ngaphandle kokukhuluma nodokotela wakho. Uma uyeka ukuthatha i-galantamine izinsuku ezimbalwa noma ngaphezulu, shayela udokotela wakho ngaphambi kokuba uqale ukuthatha i-galantamine futhi. Udokotela wakho mhlawumbe uzokutshela ukuthi uqale ngomthamo ophansi kakhulu we-galantamine futhi ukhuphule kancane umthamo wakho kumthamo obukade uwuthatha.

Ngaphambi kokuthatha isisombululo somlomo se-galantamine okokuqala ngqa, funda imiyalelo ebhaliwe eza nayo. Buza udokotela wakho noma usokhemisi ukuthi akubonise ukuthi ungasithatha kanjani isisombululo somlomo. Ukuthatha isisombululo somlomo, landela lezi zinyathelo:

  1. Vula ikepisi eliqinisekisa izingane ngokucindezela ikepisi phansi ngenkathi uliphendulela ngakwesokunxele. Susa ikepisi.
  2. Donsela i-pipette (ishubhu oyisebenzisayo ukukala umthamo we-galantamine) ngaphandle kwalo.
  3. Faka ipipette ngokuphelele ebhodleleni le-galantamine.
  4. Ngenkathi ubambe iringi engezansi ye-pipette, donsela i-pipette plunger kuye ekumaka okukhombisa umthamo odolwe ngudokotela wakho.
  5. Bamba iringi engezansi yepayipi bese ususa ipipette ebhodleleni. Qaphela ukuthi ungafaki i-plunger ngaphakathi.
  6. Lungisa ama-ounces amathathu kuya kwayi-4 (cishe inkomishi engu-1/2 [amamililitha angama-90 kuye kwayi-120]) yanoma isiphi isiphuzo esingesona esotshwala. Khipha yonke imithi kusuka kwipayipi ungene esiphuzweni ngokucindezela i-plunger yonke indlela.
  7. Faka isiphuzo kahle.
  8. Phuza yonke ingxube ngokushesha.
  9. Buyisela ikepisi lepulasitiki ebhodleleni le-galantamine bese uphendulela ikepisi ngakwesokudla ukuvala ibhodlela.
  10. Hlanza i-pipette engenalutho ngokubeka ukuphela kwayo okuvulekile engilazini yamanzi, ukhiphe i-plunger, bese uphonsa i-plunger ukuze ususe amanzi.

Lo muthi ungabekelwa okunye ukusetshenziswa; buza udokotela wakho noma usokhemisi ukuthola eminye imininingwane.


Ngaphambi kokuthatha i-galantamine,

  • Tshela udokotela kanye nosokhemisi wakho uma uxabana ne-galantamine, noma imiphi eminye imithi, noma iziphi izithako ezingasebenzi kumaphilisi e-galantamine, isixazululo, noma amaphilisi akhishwa isikhathi eside. Buza usokhemisi wakho ukuthola uhlu lwezithako ezingasebenzi.
  • Tshela udokotela wakho kanye nosokhemisi ukuthi imiphi imishanguzo kadokotela neyokungabhalisi, amavithamini, izithako zokudla okunempilo, nemikhiqizo yamakhambi oyithathayo noma ohlela ukuyithatha. Qiniseka ukuthi usho noma yikuphi okulandelayo: i-ambenonium chloride (Mytelase); i-amitriptyline (u-Elavil); imishanguzo ye-anticholinergic efana ne-atropine (Atropen, Sal-Tropine), belladonna (eDonnatal, Bellamine, Bel-Tabs, abanye); i-benztropine (Cogentin), i-biperiden (i-Akineton); clidinium (eLibrax), dicyclomine (Bentyl), glycopyrrolate (Robinul), hyoscyamine (Cytospaz-M, Levbid, Levsin), ipratropium (Atrovent, in Combivent), oxybutynin (Ditropan), procyclidine (Kemadrin), propantheine (Pro ), scopolamine (Scopace, Transderm-Scop), tiotropium (Spiriva), tolterodine (Detrol), kanye ne-trihexyphenidyl; ezinye izinto zokuvikela ezifana ne-fluconazole (i-Diflucan), i-itraconazole (i-Sporanox), i-ketoconazole (i-Nizoral), ne-voriconazole (i-Vfend); i-aspirin noma ezinye izidakamizwa ezingezona ukuvuvukala (ama-NSAID) njenge-ibuprofen (Advil, Motrin) ne-naproxen (Aleve, Naprosyn); i-bethanechol (i-Urecholine); i-cevimeline (i-Evoxac); i-cimetidine (Tagamet); i-clarithromycin (i-Biaxin, ku-Prevpac); i-digoxin (i-Lanoxin); i-fluoxetine (i-Prozac, i-Sarafem); i-fluvoxamine (i-Luvox); imithi yenhliziyo; nefazodone; i-neostigmine (Prostigmin); eminye imithi yesifo i-Alzheimer's; imishanguzo yegciwane lesandulela ngculaza (i-HIV) noma i-immunodeficiency syndrome (i-AIDS); imithi yomfutho wegazi ophakeme; i-paroxetine (Paxil); i-pyridostigmine (iMestinon); ne-quinidine (i-Quinidex). Udokotela wakho angadinga ukushintsha imithamo yemithi yakho noma akuqaphele ngokucophelela ngemiphumela emibi.
  • utshele udokotela wakho uma uke waba nesifo somoya noma esinye isifo samaphaphu; i-prostate ekhulisiwe; izilonda; ukuquleka; ukushaya kwenhliziyo okungajwayelekile; noma isifo senhliziyo, sezinso, noma sesibindi.
  • tshela udokotela wakho uma ukhulelwe, hlela ukukhulelwa, noma uncelisa. Uma ukhulelwa ngenkathi uthatha i-galantamine, shayela udokotela wakho.
  • uma uhlinzwa, kufaka phakathi ukuhlinzwa kwamazinyo, tshela udokotela noma udokotela wamazinyo ukuthi uthatha i-galantamine.
  • kufanele wazi ukuthi i-galantamine ingakwenza ukozele. Ungashayeli imoto noma usebenzise imishini uze wazi ukuthi lo muthi ukuthinta kanjani.
  • khumbula ukuthi utshwala bungangezela ukozela okubangelwa yilomuthi.

Ngaphandle kokuthi udokotela wakho akutshele ngenye indlela, qhubeka nokudla okuvamile.


Thatha umthamo ongabanjwanga ngokushesha nje lapho uwukhumbula. Kodwa-ke, uma sekuyisikhathi somthamo olandelayo, weqa umthamo ongabanjwanga bese uqhubeka neshejuli yakho ejwayelekile yokulinganisa. Ungathathi umthamo ophindwe kabili ukwenza okulahlekile.

IGalantamine ingadala imiphumela emibi. Tshela udokotela wakho uma kukhona kulezi zimpawu ezinzima noma ezingapheli:

  • isicanucanu
  • ukuhlanza
  • isifo sohudo
  • ukulahlekelwa isifiso sokudla
  • ubuhlungu besisu
  • isilungulela
  • ukuncipha komzimba
  • ukukhathala ngokweqile
  • isiyezi
  • isikhumba esiphaphathekile
  • ikhanda
  • ukuzamazama kwengxenye yomzimba wakho ongeke ukwazi ukuyilawula
  • ukudana
  • ubunzima bokulala noma ukulala
  • ikhala eligijimayo

Eminye imiphumela emibi ingaba mibi. Izimpawu ezilandelayo azivamile, kepha uma uhlangabezana nenye yazo, shayela udokotela wakho ngokushesha:

  • ubunzima bokuchama
  • igazi emchameni
  • ubuhlungu noma ukushisa ngenkathi uchama
  • isithuthwane
  • ukushaya kwenhliziyo okwehlisiwe
  • ukuquleka
  • ukuphelelwa umoya
  • indle emnyama neyokulinda
  • igazi elibomvu ezansi
  • ukuhlanza okunegazi
  • hlanza okubukeka njengezizathu zekhofi

IGalantamine ingadala eminye imiphumela emibi. Shayela udokotela wakho uma unezinkinga ezingavamile ngenkathi uthatha lo muthi.

Uma uthola imiphumela emibi kakhulu, wena noma udokotela wakho ungathumela umbiko kuhlelo lwe-Food and Drug Administration's (FDA) MedWatch Adverse Event Reporting online (http://www.fda.gov/Safety/MedWatch) noma ngocingo ( 1-800-332-1088).

Gcina le mithi esitsheni efike ngayo, ivalwe ngokuqinile, futhi lapho izingane zingafinyeleleki khona. Gcina ekamelweni lokushisa futhi kude nokushisa okweqile nomswakama (hhayi endlini yangasese).Ungafrizi.

Kubalulekile ukugcina yonke imishanguzo ingabonakali futhi ifinyeleleke ezinganeni njengoba iziqukathi eziningi (njengezingqondo zamaphilisi zamasonto onke kanye nalawo amaconsi wamehlo, okhilimu, amabala, kanye nama-inhalers) azimeleki ezinganeni futhi izingane ezincane zingazivula kalula. Ukuvikela izingane ezisencane ekufakeni ubuthi, hlala uvala amakepisi okuphepha bese ubeka umuthi endaweni ephephile - eyodwa ephezulu futhi engekho futhi engabonakali kubo futhi efinyelela kuyo. http://www.upandaway.org

Imithi engadingeki kufanele ilahlwe ngezindlela ezikhethekile zokuqinisekisa ukuthi izilwane ezifuywayo, izingane nabanye abantu abakwazi ukuzidla. Kodwa-ke, akufanele ukhiphe le mithi ethoyilethi. Esikhundleni salokho, indlela engcono kakhulu yokulahla imithi yakho ngohlelo lokubuyisa umuthi. Khuluma nosokhemisi wakho noma uthinte umnyango wangakini wokulahla udoti / wokusebenzisa kabusha ukuze ufunde ngezinhlelo zokubuyisa emphakathini wakho. Bheka iwebhusayithi yakwa-FDA's Safe Disposal of Medicines (http://goo.gl/c4Rm4p) ukuthola eminye imininingwane uma ungakwazi ukufinyelela kuhlelo lokubuyisa.

Uma kwenzeka ukweqisa ngokweqile, shayela ucingo losizo lokulawula ubuthi ku-1-800-222-1222. Imininingwane iyatholakala online ku-https: //www.poisonhelp.org/help. Uma isisulu siwile, saba nokuquleka, sinenkinga yokuphefumula, noma singakwazi ukuvuswa, shayela ngokushesha abezimo eziphuthumayo ku-911.

Izimpawu zokudlula ngokweqile zingafaka:

  • ubuthakathaka bemisipha noma ukudikiza
  • isicanucanu
  • ukuhlanza
  • amajaqamba esiswini
  • ukumunca amathe
  • amehlo anezinyembezi
  • ukwanda kokuchama
  • udinga ukuba nokunyakaza kwamathumbu
  • ukujuluka
  • ukushaya kwenhliziyo okuphuzile, okusheshayo, noma okungajwayelekile
  • ubumhlophe
  • isiyezi
  • ukuquleka
  • ukuphefumula kancane
  • ukuwa
  • ukulahlekelwa ukwazi
  • isithuthwane
  • umlomo owomile
  • ubuhlungu besifuba
  • ukusangana (ukubona izinto noma ukuzwa amazwi angekho)

Gcina wonke ama-aphoyintimenti nodokotela wakho.

Ungavumeli omunye umuntu ukuthi athathe imithi yakho. Buza usokhemisi wakho noma imiphi imibuzo onayo mayelana nokugcwalisa umuthi wakho.

Kubalulekile ukuthi ugcine uhlu olubhaliwe lwayo yonke imishanguzo oyisebenzisayo kadokotela kanye nokungabhaliswanga (ngaphezulu kokuthenga), kanye nanoma yimiphi imikhiqizo efana namavithamini, amaminerali, noma ezinye izithako zokudla. Kufanele uze nalolu hlu njalo uma uvakashela udokotela noma uma ungeniswa esibhedlela. Kubaluleke kakhulu futhi nemininingwane ebalulekile ukuthi uphathe uma kwenzeka kunezimo eziphuthumayo.

  • URazadyne® (phambilini ibitholakala njenge-Reminyl®)
  • URazadyne® ER
Kugcine ukubuyekezwa - 03/15/2020

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