I-Dipyrone

-Delile
- Yenzelwe ini
- Ungathatha kanjani
- 1. Iphilisi elilula
- 2. Ithebhulethi ye-Effervescent
- 3. Isixazululo somlomo 500 mg / mL
- 4. Isixazululo somlomo 50 mg / mL
- 5. Isengezo
- 6. Isixazululo somjovo
- Isebenza kanjani
- Imiphumela emibi engaba khona
- Ngubani ongafanele asebenzise
- Ezimweni zomkhuhlane, i-dipyrone kufanele ithathwe ngaluphi izinga lokushisa?
I-Dipyrone ngumuthi we-analgesic, antipyretic kanye ne-spasmolytic, osetshenziswa kakhulu ekwelapheni ubuhlungu nomkhuhlane, imvamisa obangelwa imikhuhlane nomkhuhlane, isibonelo.
IDipyrone ingathengwa emakhemisi ajwayelekile ngaphansi kwegama lomkhiqizo elithi Novalgina, Anador, Baralgin, Magnopyrol noma Nofebrin, ngesimo samaconsi, amaphilisi, i-suppository noma njengesisombululo somjovo, ngentengo engahluka phakathi kwama-reais ama-2 kuye kwangama-20, kuya ngokuthi isilinganiso nefomu lokwethula.
Yenzelwe ini
I-Dipyrone ikhonjisiwe ekwelapheni ubuhlungu nomkhuhlane. Imiphumela ye-analgesic ne-antipyretic ingalindelwa emaminithini angama-30 kuye kwangama-60 ngemuva kokuphathwa futhi ngokuvamile ihlala cishe amahora angama-4.
Ungathatha kanjani
Umthamo uncike kwifomu lokulinganisa elisetshenzisiwe:
1. Iphilisi elilula
Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungamaphilisi ayi-1 kuya kwangu-2 we-500 mg noma ithebhulethi elingu-1 ka-1000 mg kuze kube izikhathi ezine ngosuku. Lo muthi akufanele uhlafunwe.
2. Ithebhulethi ye-Effervescent
Ithebhulethi kufanele ichithwe uhhafu wengilazi yamanzi futhi kufanele iphuzwe ngokushesha ngemuva kokuphela kokuphela. Umthamo onconyiwe yithebhulethi elingu-1 kuze kube izikhathi ezine ngosuku.
3. Isixazululo somlomo 500 mg / mL
Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungamaconsi angama-20 kuye kwangama-40 kumthamo owodwa noma kuze kube ngamaconsi angama-40, izikhathi ezine ngosuku. Ezinganeni, umthamo kufanele uvumelane nesisindo nobudala, ngokusho kwetafula elilandelayo:
Isisindo (isilinganiso seminyaka) | Umthamo | Amaconsi |
5 kuya ku-8 kg (izinyanga ezintathu kuya kwezingu-11) | Umthamo owodwa Umthamo omkhulu | Amaconsi amabili kuya kwangu-5 20 (4 imithamo x 5 amaconsi) |
I-9 kuye ku-15 kg (iminyaka engu-1 kuye kwengu-3) | Umthamo owodwa Umthamo omkhulu | Amaconsi amathathu kuya kwayi-10 40 (amanani ama-4 x amaconsi ayi-10) |
16 kuya ku-23 kg (iminyaka emi-4 kuye kwengu-6) | Umthamo owodwa Umthamo omkhulu | Amaconsi ama-5 kuye kwayi-15 60 (imithamo emi-4 x amaconsi angu-15) |
24 kuya ku-30 kg (iminyaka engu-7 kuya kwengu-9) | Umthamo owodwa Umthamo omkhulu | Amaconsi angu-8 kuya kwangu-20 80 (amanani ama-4 x amaconsi angu-20) |
31 kuya ku-45 kg (iminyaka eyi-10 kuye kwengu-12) | Umthamo owodwa Umthamo omkhulu | Amaconsi ayi-10 kuye kwangama-30 I-120 (imithamo emi-4 x 30 amaconsi) |
46 kuya ku-53 kg (iminyaka engu-13 kuya kwengu-14) | Umthamo owodwa Umthamo omkhulu | 15 kuya ku-35 amaconsi 140 (4 kuthatha x 35 amaconsi) |
Izingane ezingaphansi kwezinyanga ezintathu ubudala noma ezinesisindo esingaphansi kuka-5 kg akufanele ziphathwe ngeDipyrone.
4. Isixazululo somlomo 50 mg / mL
Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungama-10 kuye kwangama-20 mL, ngomthamo owodwa noma kufika kuma-20 mL, amahlandla ama-4 ngosuku. Ezinganeni, umthamo kufanele unikezwe ngokwesisindo nobudala, ngokusho kwetafula elingezansi:
Isisindo (isilinganiso seminyaka) | Umthamo | Isixazululo somlomo (ku-mL) |
5 kuya ku-8 kg (izinyanga ezintathu kuya kwezingu-11) | Umthamo owodwa Umthamo omkhulu | 1.25 kuye ku-2,5 10 (amanani ama-4 x 2.5 mL) |
I-9 kuye ku-15 kg (iminyaka engu-1 kuye kwengu-3) | Umthamo owodwa Umthamo omkhulu | 2.5 kuye ku-5 20 (imithamo emi-4 x 5 ml) |
16 kuya ku-23 kg (iminyaka emi-4 kuye kwengu-6) | Umthamo owodwa Umthamo omkhulu | 3.75 kuye ku-7.5 30 (amanani ama-4 x 7.5 mL) |
24 kuya ku-30 kg (iminyaka engu-7 kuya kwengu-9) | Umthamo owodwa Umthamo omkhulu | 5 kuye ku-10 40 (4 x 10 mL amasokhethi) |
31 kuya ku-45 kg (iminyaka eyi-10 kuye kwengu-12) | Umthamo owodwa Umthamo omkhulu | 7.5 kuya ku-15 60 (amasokhethi amane x 15 mL) |
46 kuya ku-53 kg (iminyaka engu-13 kuya kwengu-14) | Umthamo owodwa Umthamo omkhulu | 8.75 kuya ku-17.5 70 (amasokhethi amane x 17.5 ml) |
Izingane ezingaphansi kwezinyanga ezintathu ubudala noma ezinesisindo esingaphansi kuka-5 kg akufanele ziphathwe ngeDipyrone.
5. Isengezo
Ama-suppositories kufanele asetshenziswe ngokweqile, ngokulandelayo:
- Njalo gcina okufakwayo kwe-suppository endaweni epholile;
- Uma ama-suppositories ethanjiswa ukushisa, ukufakwa kwe-aluminium kufanele kucwiliswe imizuzwana embalwa emanzini e-ice ukubabuyisela ekuvumelaneni kwabo kwasekuqaleni;
- Ukulandela ukufakwa kwephakeji ye-aluminium, kuphela i-suppository ezosetshenziswa okufanele ivezwe;
- Ngaphambi kokufaka i-suppository, kufanele ugeze izandla zakho kahle futhi, uma kungenzeka, uzifake amagciwane ngotshwala;
- Ngomunwe wakho wesithupha nowenkomba, hambisa izinqa zakho ngaphandle bese ufaka i-suppository ku-orifice yangemuva bese ucindezela ngobumnene izinqe elilodwa ulibhekise komunye imizuzwana embalwa ukuvimbela ukuthi i-suppository ingabuyi.
Umthamo onconywayo yi-1 suppository, kuze kube izikhathi ezine ngosuku. Uma umphumela womthamo owodwa unganele noma ngemuva kokuncipha kwe-analgesic, umthamo ungaphindwa maqondana ne-posology kanye nomthamo omkhulu wansuku zonke.
6. Isixazululo somjovo
I-dipyrone ejojoweyo ingalawulwa ngemithambo yegazi noma nge-intramuscularly, lapho umuntu elele phansi nangaphansi kokuqondiswa ngudokotela. Ngaphezu kwalokho, ukuphathwa ngemithambo kufanele kuhambe kancane, ngesilinganiso sokumnika esingadluli kuma-500 mg we-dipyrone ngomzuzu, ukuvimbela ukusabela kwe-hypotensive.
Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungu-2 kuye ku-5 ml ngomthamo owodwa, kuze kufike kumthamo omkhulu wansuku zonke we-10 mL. Ezinganeni nasezinsaneni, umthamo onconyiwe uncike esisindweni, njengoba kukhonjisiwe etafuleni elilandelayo:
Isisindo | Umthamo (ku-mL) |
Izinsana ezisuka ku-5 kuye ku-8 kg | 0.1 - 0.2 ml |
Izingane ezisuka ku-9 kuye ku-15 kg | 0.2 - 0.5 ml |
Izingane ezisuka ku-16 kuye ku-23 kg | 0.3 - 0.8 mL |
Izingane ezisuka kuma-24 kuye kuma-30 kg | 0.4 - 1.0 ml |
Izingane ezisuka ku-31 kuye ku-45 kg | 0.5 - 1.5 ml |
Izingane ezisuka kuma-46 kuye kuma-53 kg | 0.8 - 1.8 ml |
Uma ukuphathwa kwabazali kwe-dipyrone kucatshangelwa ezinganeni ezisuka ku-5 kuye ku-8 kg, kufanele kusetshenziswe umzila we-intramuscular kuphela.
Isebenza kanjani
I-Dipyrone yinto enemiphumela ye-analgesic, antipyretic kanye ne-spasmolytic. I-Dipyrone iyi-prodrug, okusho ukuthi isebenza kuphela ngemuva kokufakwa nokufakwa emzimbeni.
Olunye ucwaningo luphakamisa ukuthi ama-metabolites asebenzayo e-dipyrone enza ngokuvimbela ama-enzyme cyclooxygenase (COX-1, COX-2 kanye ne-COX-3), evimbela ukuhlanganiswa kwama-prostaglandin, okungcono ohlelweni lwezinzwa oluphakathi nokwenza i-receptors yezinhlungu zangaphandle zingasebenzi. umsebenzi nge-nitric oxide-cGMP ku-receptor yezinhlungu.
Imiphumela emibi engaba khona
Imiphumela emibi yeDipyrone ifaka phakathi isifuba, umfutho wegazi ophansi, izinso nezinkinga zomchamo, ukuphazamiseka kwemithambo yegazi kanye nokwaliwa okukhulu.
Ngubani ongafanele asebenzise
I-Dipyrone iyaphikiswa ekukhulelweni, ekunceliseni ibele nakubantu abanokungezwani komzimba ne-sodium dipyrone noma enye yezinhlobo zefomula, i-asthma, i-acute intermittent liver porphyria kanye ne-congenital glucose-6-phosphate dehydrogenase.
Iziguli ezenze i-bronchospasm noma okunye ukusabela kwe-anaphylactic nge-analgesics, njenge-salicylates, i-paracetamol, i-diclofenac, i-ibuprofen, i-indomethacin ne-naproxen, nayo akufanele ithathe i-sodium dipyrone.
Ezimweni zomkhuhlane, i-dipyrone kufanele ithathwe ngaluphi izinga lokushisa?
Umkhuhlane uphawu oludinga ukulawulwa kuphela uma lubanga ukungaphatheki kahle noma lubeka engcupheni isimo somuntu jikelele. Ngakho-ke, i-dipyrone kufanele isetshenziswe kuphela kulezi zimo noma uma ikhonjiswa ngudokotela.