Umlobi: Frank Hunt
Usuku Lokudalwa: 16 Hamba 2021
Ukuvuselela Usuku: 5 Epreli 2025
Anonim
DIPYRONE 2.0
Ividiyo: DIPYRONE 2.0

-Delile

I-Dipyrone ngumuthi we-analgesic, antipyretic kanye ne-spasmolytic, osetshenziswa kakhulu ekwelapheni ubuhlungu nomkhuhlane, imvamisa obangelwa imikhuhlane nomkhuhlane, isibonelo.

IDipyrone ingathengwa emakhemisi ajwayelekile ngaphansi kwegama lomkhiqizo elithi Novalgina, Anador, Baralgin, Magnopyrol noma Nofebrin, ngesimo samaconsi, amaphilisi, i-suppository noma njengesisombululo somjovo, ngentengo engahluka phakathi kwama-reais ama-2 kuye kwangama-20, kuya ngokuthi isilinganiso nefomu lokwethula.

Yenzelwe ini

I-Dipyrone ikhonjisiwe ekwelapheni ubuhlungu nomkhuhlane. Imiphumela ye-analgesic ne-antipyretic ingalindelwa emaminithini angama-30 kuye kwangama-60 ngemuva kokuphathwa futhi ngokuvamile ihlala cishe amahora angama-4.

Ungathatha kanjani

Umthamo uncike kwifomu lokulinganisa elisetshenzisiwe:

1. Iphilisi elilula

Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungamaphilisi ayi-1 kuya kwangu-2 we-500 mg noma ithebhulethi elingu-1 ka-1000 mg kuze kube izikhathi ezine ngosuku. Lo muthi akufanele uhlafunwe.


2. Ithebhulethi ye-Effervescent

Ithebhulethi kufanele ichithwe uhhafu wengilazi yamanzi futhi kufanele iphuzwe ngokushesha ngemuva kokuphela kokuphela. Umthamo onconyiwe yithebhulethi elingu-1 kuze kube izikhathi ezine ngosuku.

3. Isixazululo somlomo 500 mg / mL

Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungamaconsi angama-20 kuye kwangama-40 kumthamo owodwa noma kuze kube ngamaconsi angama-40, izikhathi ezine ngosuku. Ezinganeni, umthamo kufanele uvumelane nesisindo nobudala, ngokusho kwetafula elilandelayo:

Isisindo (isilinganiso seminyaka)UmthamoAmaconsi 
5 kuya ku-8 kg (izinyanga ezintathu kuya kwezingu-11)

Umthamo owodwa

Umthamo omkhulu

Amaconsi amabili kuya kwangu-5

20 (4 imithamo x 5 amaconsi)

I-9 kuye ku-15 kg (iminyaka engu-1 kuye kwengu-3)

Umthamo owodwa

Umthamo omkhulu

Amaconsi amathathu kuya kwayi-10

40 (amanani ama-4 x amaconsi ayi-10)

16 kuya ku-23 kg (iminyaka emi-4 kuye kwengu-6)

Umthamo owodwa

Umthamo omkhulu

Amaconsi ama-5 kuye kwayi-15

60 (imithamo emi-4 x amaconsi angu-15)


24 kuya ku-30 ​​kg (iminyaka engu-7 kuya kwengu-9)

Umthamo owodwa

Umthamo omkhulu

Amaconsi angu-8 kuya kwangu-20

80 (amanani ama-4 x amaconsi angu-20)

31 kuya ku-45 kg (iminyaka eyi-10 kuye kwengu-12)

Umthamo owodwa

Umthamo omkhulu

Amaconsi ayi-10 kuye kwangama-30

I-120 (imithamo emi-4 x 30 amaconsi)

46 kuya ku-53 kg (iminyaka engu-13 kuya kwengu-14)

Umthamo owodwa

Umthamo omkhulu

15 kuya ku-35 amaconsi

140 (4 kuthatha x 35 amaconsi)

Izingane ezingaphansi kwezinyanga ezintathu ubudala noma ezinesisindo esingaphansi kuka-5 kg ​​akufanele ziphathwe ngeDipyrone.

4. Isixazululo somlomo 50 mg / mL

Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungama-10 kuye kwangama-20 mL, ngomthamo owodwa noma kufika kuma-20 mL, amahlandla ama-4 ngosuku. Ezinganeni, umthamo kufanele unikezwe ngokwesisindo nobudala, ngokusho kwetafula elingezansi:

Isisindo (isilinganiso seminyaka)UmthamoIsixazululo somlomo (ku-mL)

5 kuya ku-8 kg (izinyanga ezintathu kuya kwezingu-11)


Umthamo owodwa

Umthamo omkhulu

1.25 kuye ku-2,5

10 (amanani ama-4 x 2.5 mL)

I-9 kuye ku-15 kg (iminyaka engu-1 kuye kwengu-3)

Umthamo owodwa

Umthamo omkhulu

2.5 kuye ku-5

20 (imithamo emi-4 x 5 ml)

16 kuya ku-23 kg (iminyaka emi-4 kuye kwengu-6)

Umthamo owodwa

Umthamo omkhulu

3.75 kuye ku-7.5

30 (amanani ama-4 x 7.5 mL)

24 kuya ku-30 ​​kg (iminyaka engu-7 kuya kwengu-9)

Umthamo owodwa

Umthamo omkhulu

5 kuye ku-10

40 (4 x 10 mL amasokhethi)

31 kuya ku-45 kg (iminyaka eyi-10 kuye kwengu-12)

Umthamo owodwa

Umthamo omkhulu

7.5 kuya ku-15

60 (amasokhethi amane x 15 mL)

46 kuya ku-53 kg (iminyaka engu-13 kuya kwengu-14)

Umthamo owodwa

Umthamo omkhulu

8.75 kuya ku-17.5

70 (amasokhethi amane x 17.5 ml)

Izingane ezingaphansi kwezinyanga ezintathu ubudala noma ezinesisindo esingaphansi kuka-5 kg ​​akufanele ziphathwe ngeDipyrone.

5. Isengezo

Ama-suppositories kufanele asetshenziswe ngokweqile, ngokulandelayo:

  1. Njalo gcina okufakwayo kwe-suppository endaweni epholile;
  2. Uma ama-suppositories ethanjiswa ukushisa, ukufakwa kwe-aluminium kufanele kucwiliswe imizuzwana embalwa emanzini e-ice ukubabuyisela ekuvumelaneni kwabo kwasekuqaleni;
  3. Ukulandela ukufakwa kwephakeji ye-aluminium, kuphela i-suppository ezosetshenziswa okufanele ivezwe;
  4. Ngaphambi kokufaka i-suppository, kufanele ugeze izandla zakho kahle futhi, uma kungenzeka, uzifake amagciwane ngotshwala;
  5. Ngomunwe wakho wesithupha nowenkomba, hambisa izinqa zakho ngaphandle bese ufaka i-suppository ku-orifice yangemuva bese ucindezela ngobumnene izinqe elilodwa ulibhekise komunye imizuzwana embalwa ukuvimbela ukuthi i-suppository ingabuyi.

Umthamo onconywayo yi-1 suppository, kuze kube izikhathi ezine ngosuku. Uma umphumela womthamo owodwa unganele noma ngemuva kokuncipha kwe-analgesic, umthamo ungaphindwa maqondana ne-posology kanye nomthamo omkhulu wansuku zonke.

6. Isixazululo somjovo

I-dipyrone ejojoweyo ingalawulwa ngemithambo yegazi noma nge-intramuscularly, lapho umuntu elele phansi nangaphansi kokuqondiswa ngudokotela. Ngaphezu kwalokho, ukuphathwa ngemithambo kufanele kuhambe kancane, ngesilinganiso sokumnika esingadluli kuma-500 mg we-dipyrone ngomzuzu, ukuvimbela ukusabela kwe-hypotensive.

Umthamo onconyelwe abantu abadala nentsha engaphezu kweminyaka engu-15 ungu-2 kuye ku-5 ml ngomthamo owodwa, kuze kufike kumthamo omkhulu wansuku zonke we-10 mL. Ezinganeni nasezinsaneni, umthamo onconyiwe uncike esisindweni, njengoba kukhonjisiwe etafuleni elilandelayo:

IsisindoUmthamo (ku-mL)
Izinsana ezisuka ku-5 kuye ku-8 kg0.1 - 0.2 ml
Izingane ezisuka ku-9 kuye ku-15 kg0.2 - 0.5 ml
Izingane ezisuka ku-16 kuye ku-23 kg0.3 - 0.8 mL
Izingane ezisuka kuma-24 kuye kuma-30 kg0.4 - 1.0 ml
Izingane ezisuka ku-31 kuye ku-45 kg0.5 - 1.5 ml
Izingane ezisuka kuma-46 kuye kuma-53 kg0.8 - 1.8 ml

Uma ukuphathwa kwabazali kwe-dipyrone kucatshangelwa ezinganeni ezisuka ku-5 kuye ku-8 kg, kufanele kusetshenziswe umzila we-intramuscular kuphela.

Isebenza kanjani

I-Dipyrone yinto enemiphumela ye-analgesic, antipyretic kanye ne-spasmolytic. I-Dipyrone iyi-prodrug, okusho ukuthi isebenza kuphela ngemuva kokufakwa nokufakwa emzimbeni.

Olunye ucwaningo luphakamisa ukuthi ama-metabolites asebenzayo e-dipyrone enza ngokuvimbela ama-enzyme cyclooxygenase (COX-1, COX-2 kanye ne-COX-3), evimbela ukuhlanganiswa kwama-prostaglandin, okungcono ohlelweni lwezinzwa oluphakathi nokwenza i-receptors yezinhlungu zangaphandle zingasebenzi. umsebenzi nge-nitric oxide-cGMP ku-receptor yezinhlungu.

Imiphumela emibi engaba khona

Imiphumela emibi yeDipyrone ifaka phakathi isifuba, umfutho wegazi ophansi, izinso nezinkinga zomchamo, ukuphazamiseka kwemithambo yegazi kanye nokwaliwa okukhulu.

Ngubani ongafanele asebenzise

I-Dipyrone iyaphikiswa ekukhulelweni, ekunceliseni ibele nakubantu abanokungezwani komzimba ne-sodium dipyrone noma enye yezinhlobo zefomula, i-asthma, i-acute intermittent liver porphyria kanye ne-congenital glucose-6-phosphate dehydrogenase.

Iziguli ezenze i-bronchospasm noma okunye ukusabela kwe-anaphylactic nge-analgesics, njenge-salicylates, i-paracetamol, i-diclofenac, i-ibuprofen, i-indomethacin ne-naproxen, nayo akufanele ithathe i-sodium dipyrone.

Ezimweni zomkhuhlane, i-dipyrone kufanele ithathwe ngaluphi izinga lokushisa?

Umkhuhlane uphawu oludinga ukulawulwa kuphela uma lubanga ukungaphatheki kahle noma lubeka engcupheni isimo somuntu jikelele. Ngakho-ke, i-dipyrone kufanele isetshenziswe kuphela kulezi zimo noma uma ikhonjiswa ngudokotela.

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